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Slide Lecture Programs
2007 Core Curriculum
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Contemporary Management of Cardiometabolic Risk
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May 15, 2007
Table of Contents - 105 slides
No.
Title
1
Contemporary Management of Cardiometabolic Risk
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2
A continuing epidemic: 2 of 3 US adults are overweight or obese
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3
Parallel epidemics of diabetes and obesity
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4
Defining cardiometabolic risk
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5
Associations of adiposity with CVD
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6
Adiposity predicts mortality
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7
Adiposity associated with premature MI
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8
Majority of patients undergoing PCI are overweight or obese
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9
Adverse consequences of chronic adiposity and ectopic fat
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10
Epicardial adipose tissue may be increased in visceral obesity
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11
Adiposity in the development of NASH
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12
Visceral vs subcutaneous adiposity
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13
Neutral effect of liposuction on cardiometabolic risk factors
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14
Central adiposity: Better marker of CVD than BMI
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15
A new vital sign: Waist circumference
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16
Continued burden of disease
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17
Adiposity in CVD
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18
Role of adipose tissue in atherogenesis
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19
Elevated FFA contribute to hypertension, dyslipidemia, and insulin resistance
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20
Energy homeostasis is linked to immune balance
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21
Weight gain induces inflammatory changes in adipose tissue
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22
Adipose tissue: An endocrine organ
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23
Adiponectin associated with decreased risk of MI
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24
Beneficial associations of adiponectin
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25
Low adiponectin in visceral adiposity
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26
Even moderate weight loss may improve cardiometabolic risk
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27
Summary
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28
The Endocannabinoid System
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29
Cannabinoid classification with selected examples
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30
ECS: Widely distributed with multiple cardiometabolic effects
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31
Potential therapeutic implications of CB
1
receptor blockade
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32
Circulating 2-AG elevated in persons with visceral vs sc adiposity
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33
CB
1
receptor blockade blunts overeating in rats
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34
CB
1
receptor blockade: Weight reduction independent of food intake in obese mice
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35
CB
1
receptor blockade modulates adipocyte function in mice
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36
CB
1
receptors modulate liver lipogenesis in mice
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37
CB
1
receptor blockade increases skeletal muscle glucose uptake in obese mice
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38
CB
1
receptor blockade and mood: Range of effects observed in animal models
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39
Endocannabinoid system overview
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40
Managing Cardiometabolic Risk
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41
NHLBI guidelines: Adiposity assessment
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42
BMI classifications
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43
Measuring waist circumference
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44
Diagnostic criteria for metabolic syndrome
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45
NHLBI guidelines: Weight loss goals
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46
Guide to adiposity management
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47
NHLBI guidelines: Lifestyle modification
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48
Some moderate-intensity physical activities
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49
3-Week diet + exercise regimen yields favorable metabolic changes
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50
Physical activity may reduce CV and all-cause mortality
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51
Lifestyle modification associated with diabetes prevention
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52
DPP: Benefit of diet + exercise or metformin on diabetes prevention in at-risk patients
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53
Popular dietary programs: Effective yet difficult to maintain
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54
Look AHEAD: Study design
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55
NHLBI guidelines: Pharmacologic therapy
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56
Pharmacologic weight management options
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57
Efficacy of orlistat as adjunct to lifestyle modification
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58
Efficacy of sibutramine as adjunct to lifestyle modification
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59
Effects of sibutramine and lifestyle modification on cardiometabolic risk factors
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60
SCOUT: Study design
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61
NHLBI guidelines: Weight loss surgery
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62
SOS: Bariatric surgery-associated improvements in cardiometabolic risk
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63
Improved Framingham risk score following bariatric surgery
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64
Clinical evaluation of CB
1
receptor blockade
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65
Rimonabant In Obesity (RIO) program
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66
RIO program: Improved cardiometabolic risk factors at 1 year
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67
RIO program: Decreased metabolic syndrome incidence
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68
RIO program: Safety and tolerability
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69
RIO program: No significant effect on mood
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70
RIO program: Mood at 1 year
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71
RIO clinical trial program efficacy summary
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72
SERENADE: Study design
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73
SERENADE: Change in A1C at 6 months
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74
Summary
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75
Ongoing trials with rimonabant in abdominal adiposity
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76
Current and emerging pharmacologic combinations for treating cardiometabolic risk
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77
Managing cardiometabolic risk
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78
Data Supplement
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79
RIO-Europe: Study design
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80
RIO-Europe: Treatment effect on weight and waist circumference
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81
RIO-Europe: Treatment effect on lipids
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82
RIO-Europe: Adverse events
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83
RIO-Lipids: Study design
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84
RIO-Lipids: Treatment effect on weight and WC
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85
RIO-Lipids: Treatment effect on lipids
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86
RIO-Lipids: Rimonabant weight-independent effect on adiponectin
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87
RIO-Lipids: Adverse events
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88
RIO-Diabetes: Study design
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89
RIO-Diabetes: Treatment effect on weight and waist circumference
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90
RIO-Diabetes: Treatment effect on lipids
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91
RIO-Diabetes: Treatment effect on glucose metabolism
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92
RIO-Diabetes: Adverse events
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93
RIO-North America: Study design
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94
RIO-North America: Weight change by treatment assignment
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95
RIO-North America: Waist circumference by treatment assignment
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96
RIO-North America: Treatment effect on lipids at 1 year
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97
RIO-North America: Weight-independent and weight-dependent effects on lipids
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98
RIO-North America: Weight-independent and weight-dependent effects on insulin and IR
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99
RIO-North America: Adverse events
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100
RIO-North America: Adverse events, cont'd
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101
Obesity program depression-related events: Overall incidences
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102
Completed phase 2 and 3 studies as of March 2007: All suicidality-related events
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103
Rimonabant clinical safety: Summary
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104
ACOMPLIA: European product information
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105
ACOMPLIA: European product information, cont'd
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